Pharmacology-14 Opioid Analgesics

  1. Strong Agonists Fentanyl
    Duragesic Pain High affinity for Mu receptors Respiratory depression, constipation, abuse
  2. Strong Agonists Hydromorphone
    Dilaudid Pain High affinity for Mu receptors Respiratory depression, constipation, abuse
  3. Strong Agonists Meperidine
    Demoral Pain High affinity for Mu receptors Respiratory depression, constipation, abuse
  4. Strong Agonists Methadone
    Dolophine, Methadose Pain High affinity for Mu receptors Respiratory depression, constipation, abuse
  5. Strong Agonists Morphine
    Roxanol, Statex Pain High affinity for Mu receptors Respiratory depression, constipation, abuse
  6. Mild-to-Moderate Agonists Codeine
    Pain Not as high affinity to opioid receptors. Constipation, less risk of respiratory depression.
  7. Mild-to-Moderate Agonists Hydrocodone
    Hycodan Pain Not as high affinity to opioid receptors. Constipation, less risk of respiratory depression.
  8. Mild-to-Moderate Agonists Oxycodone
    Oxycontin Pain Not as high affinity to opioid receptors. Constipation, less risk of respiratory depression.
  9. Mild-to-Moderate Agonists Propoxyphene
    Darvon, Darvocet Pain Not as high affinity to opioid receptors. Constipation, less risk of respiratory depression.
  10. Mixed Agonist-Antagonist Butophanol
    Stadol Pain, treating opioid addictions Partially activates mu receptors, antagonist to kappa Hallucinations
  11. Mixed Agonist-Antagonist Buprenorphine
    Buprenex Pain, treating opioid addictions Partially activates mu receptors, antagonist to kappa Hallucinations
  12. Mixed Agonist-Antagonist Nalbuphrine
    Nubain Pain, treating opioid addictions Partially activates mu receptors, antagonist to kappa Hallucinations
  13. Mixed Agonist-Antagonist Pentazocine
    Talwin Pain, treating opioid addictions Partially activates mu receptors, antagonist to kappa Hallucinations
  14. Antagonists Nalmefene
    Revex Not for pain,Opioid overdose and addiction Block all opioid receptors, especially mu. Displace opioid agonists Reverse respiratory depression in 1-2 minutes
  15. Antagonists Naloxone
    Narcan Not for pain,Opioid overdose and addiction Block all opioid receptors, especially mu. Displace opioid agonists Reverse respiratory depression in 1-2 minutes
  16. Antagonists Naltrexone
    ReVia Not for pain,Opioid overdose and addiction Block all opioid receptors, especially mu. Displace opioid agonists Reverse respiratory depression in 1-2 minutes
Author
Kalanzo
ID
67240
Card Set
Pharmacology-14 Opioid Analgesics
Description
Pharmacology-14 Opioid Analgesics
Updated