Adrenergic Agonists and Antagonists

  1. primary nervous system
    CNS
  2. The CNS consists of ________ and ________.
    brain, spinal cord
  3. The peripheral nervous system (PNS), located outside the brain and spinal cord, is made up of two divisions:
    • 1. the autonomic
    • 2. the somatic
  4. The autonomic nervous system (ANS), also called the ___________, acts on smooth muscles and glands.
    visceral system
  5. Functions of ANS
    control and regulation of the heart, respiratory system, gastrointestinal tract, bladder, eyes, and glands
  6. The ANS is an involuntary nervous system over which we have little or no control. True or False?
    True
  7. _______________ is a voluntary system that innervates skeletal muscles, over which there is control.
    Somatic nervous system (SNS)
  8. Two set of neurons in autonomic component of PNS
    • Afferent (Sensory neurons)
    • Efferent (Motor neurons)
  9. The efferent pathways in the ANS are divided into two branches. What are these?
    • 1. Sympathetic Nerve
    • 2. Parasympathetic Nerve
  10. Sympathetic nerve is also called the _________________.
    adrenergic system
  11. _____________ is the neurotransmitter that innervates smooth muscles.
    Norepinephrine
  12. Adrenergic receptor organ cells are of four types:
    • Alpha1
    • Alpha2
    • Beta1
    • Beta2
  13. The sympathetic and parasympathetic nervous systems act on the same
    organs but produce opposite responses to provide homeostasis (balance). True or False?
    True
  14. Drugs that stimulate the sympathetic nervous system
    • adrenergic agonists
    • adrenergics
    • sympathomimetics
  15. When __________ receptors in vascular tissues (vessels) of muscles are
    stimulated, the arterioles and venules constricts; this increase peripheral resistance and blood return to the heart, circulation improves, and blood pressure is increased. When too much stimulation occurs, blood flow decreased to the vital organs.
    Alpha1
  16. ______receptor are in the postganglionic sympathetic nerve endings, when stimulated, they inhibit the release of norepinephrine, which leads to a decrease in vasoconstriction. This results in vasodilation and a decrease in blood pressure.
    Alpha 2
  17. Receptors are located primarily in the heart but are also found in the
    kidneys. Stimulation of the this receptor increases myocardial contractility and heart rate.
    Beta 1
  18. __________ receptors are found mostly in the smooth muscle of the lung and GI tract, the liver, and the uterine muscle.
    Beta 2
  19. Other adrenergic receptor is _____________ and are located in the renal,
    mesenteric, coronary, and cerebral arteries. When these receptor are
    stimulated, the vessels dilate and blood flow increases. Only dopamine can activate this receptor.
    dopaminergic
  20. After the neurotransmitter (e.g., norepinephrine) has performed its function, the action must be stopped to prevent prolonging the effect. Transmitters are inactivated by:
    • (1) reuptake of the transmitter back into the neuron (nerve cell terminal),
    • (2) enzymatic transformation or degradation,
    • (3) diffusion away from the receptor.
  21. The two enzymes that inactivate norepinephrine are:
    • (1) monoamine oxidase (MAO), which is inside the neuron; and
    • (2) catechol-O-methyltransferase (COMT), which is outside of the neuron.
  22. (Classification of Sympathomimetic) directly stimulate the adrenergic receptor (e.g., epinephrine or norepinephrine)
    Direct-acting sympathomimetics
  23. (Classification of Sympathomimetic)  stimulate the release of norepinephrine from the terminal nerve endings (e.g., amphetamine)
    Indirect-acting sympathomimetics
  24. (Classification of Sympathomimetic) (both direct and indirect-acting), which stimulate the adrenergic receptor sites and stimulate the release of norepinephrine from the terminal nerve endings (e.g., ephedrine)
    Mixed-acting sympathomimetics
  25. ________________  is an example of a mixed-acting sympathomimetic.
    This drug acts indirectly by stimulating the release of norepinephrine from the nerve terminals and acts directly on the alpha1 and beta1 receptors; like epinephrine, increases heart rate
    Pseudoephedrine
  26. Pseudoephedrine is helpful to relieve nasal and sinus congestion without rebound congestion. True or False?
    True
Author
raine
ID
363249
Card Set
Adrenergic Agonists and Antagonists
Description
Updated