Med Chem quiz 5

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Sotalol/Betapace
- Ethanolamine B-blocker
- 0% protein bound
Propranolol/Inderal
- Non-selective B-blocker
- Lipid soluble
- Treat pheochromocytoma, at low dose stage fright.
- PTSD and Infantile Hemangiomas
Timolol/Blocarden
- Non-selective B-blocker
- Treat MI Migraine prophylaxis
Penbutolol Sulfate/Levatol
- non-selective B-blocker
- Used when a B-blocker is needed but you dont want to slow down the heart.
Nadolol/Corgard
- non-selective B-blocker
- dosage needs reduced in renal failure
Pindolol/Visken
- non-selective B-blocker
- Provides less resting bradycardia
Carteolol/cartol
- non-selective B-blocker
- Has less resting brady effects
Atenolol/Tenormin
- B1-blockern
- At high dose you lose selectivity
Metoprolol/Lopressor
- B1-blocker
- Used to prevent cardiac remodeling
- Avoid the extended release form for presergical treatment
Bisprolol/ Zebeta
- B1-blocker
- Treat hypertension
- 50% renally excreted unchanged
Betaxolol/Kerlane
- B1-blocker
- 80% excreted in urine
- Starting dosage for elderly is 5mg
Esmolol/Brevibloc
- B1-blocker
- Treat Supraventricular tachy
- Extreme metabolism by esterases in RBC
- Incompatable with sodium bicarb
Acebutolol/Sectral
- B1-blocker
- Has less resting brady
- Treat ventricular arrhythmias
Nebivolol/Bystolic

New B1 that also modulates nitric oxide system (increase)
Labetalol
- Non-selective B and A blocker
- Treat Clonidine withdrawl
- Not compatable in basic solutions
Carvedilol
- A and B blocker
- Prodrug
- Treat essential hyper
- Metabolite is 14x stronger b blocker
- First to show pharmacogenomic factors
Prazosin/Minipress
- selective A1
- Treat BPH and Hyper
Trazosin
- A1 selective
- Treat BPH
- First dose causes postural hypotension
Alfuzosin
- Non-steroidal for BPH
- Selective blocker of SM A1 receptors
- Possible QT
Silodosin/Rapaflo
- Non-steroidal for BPH
- More selective
- No QT
Doxazosin
- Selective A1
- First dose hypo
Tamsulosin
- A1 selective (38 fold)
- One of themost popular
- Sulfa Allergy
Methyldopate and Methyldopa

Centrally acting anti-adrenergic
Clonidine/Catapres
- Centrally acting anti-adrenergic
- Treat ulcerative colitis
- Severe rebound hyper possible
Guanabenz/Wytensin
- Centrally acting anti-adrenergic
- Rarely used
Guanfacine
- Centrally acting anti-adrenergic
- Rarely used
Reserpine
- Agent that depletes neurotransmitter stores
- Depletes catacholamines
Guanadrel/Hylorel
- Depletes catacholamines
- Treat hyper not responding to thiazides
Mecamylamine
- Depletes catachol
- Not common
- Dose determined by trial and error
Guanethidine
- Depletes catachol
- Inhibits the release of norepi
Cleviprex
- Ca blocker
- Contra in soy/egg allergy
- Injectable Emulsion
Sodium Diazoxide/HyperStat
- Potassium Channel Blocker for emergency hyper
- Also treats Hyper insulinism
- Not effective against Pheochromo
Fenoldopam
- Dopamine agonist for hyper emergency
- Used short term

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75ford

176639

Card Set

Med Chem quiz 5

Description

Med Chem quiz 5

Updated

2012-10-10T00:05:38Z

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