Keefe Drugs-A.txt

  1. Mixed Agonist
    • Epinephrine
    • A1,A2,B1,B2
  2. Mixed Agonist
    • Norepinephrine
    • A1,A2,B1,B2
    • B1>>B2

    • Mixed Agonist
    • Dopamine
    • DA>A>B
    • Dose dependant

    • A-1 Agonist
    • Phenylephrine
  3. A-1 Agonist
    Midodrine
  4. A-2 Agonist
    Brimonidine
  5. B1/B2 Agonist
    Isoproterenol
  6. B-2 Agonist
    Albuterol
  7. B-2 Agonist
    Levalbuterol
  8. B-2 Agonist
    Terbutaline
  9. B-2 Agonist
    Formoterol
  10. A/B Agonist
    • Dobutamine
    • A and B, but B1 predominates
  11. A/B Agonist
    • Ephedrine
    • A and B directly, indirectly by releasing NE
  12. A/B Agonist
    • Pseudoephedrine
    • A and B directly, indirectly by releasing NE
  13. Dopamine Agonist
    • Fenoldopam
    • D1
  14. Indirect Agonist
    • Cocaine
    • Blocks NET
  15. Indirect Agonist
    • Methylphenidate
    • Blocks NET and DAT
  16. Indirect Agonist
    • Tyramine
    • Releases NE from storage vesicles
  17. A1/A2 Antagonist
    • Phenoxybenzamine
    • Irreversible
  18. A1/A2 Antagonist
    • Phentolamine
    • Competitive
  19. A-1 Antagonist
    Doxazosin
  20. A-1 Antagonist
    Terazosin
  21. A-1 Antagonist
    • Tamsulosin
    • A1a selective
  22. B1/B2 Antagonist
    Propranolol
  23. B1/B2 Antagonist
    Nadolol
  24. B1/B2 Antagonist
    Timolol
  25. B-1 Antagonist
    Metoprolol
  26. B-1 Antagonist
    Atenolol
  27. B-1 Antagonist
    Esmolol
  28. B-1 Antagonist
    Betazolol
  29. Mixed A1/B Antagonist
    Carvedilol
  30. NE Depletion
    Reserpine
  31. A-2 Agonist
    Clonidine
Author
jilbear1
ID
172292
Card Set
Keefe Drugs-A.txt
Description
Drug/Receptor
Updated