ADR exam 1

  1. Beta-Blockers (2D6 substrates):
         carvedilol
         metoprolol
         nebivolol
         propranolol
         timolol
    CYP2D6 inhibitors
  2. Anxiolytics/Hypnotics:
         benzodiazepines
         buspirone
         clorazepate
    CYP3A4 inhibitors
  3. Azole antifungals:
         itraconazole
         ketoconazole
         posaconazole
         voriconazole
    Enzyme inducers
  4. Antiarrhythmics:
         amiodarone
         disopyramide
         dronedarone
         quinidine
    • CYP3A4 inhibitors
    • Enzyme inducers
  5. Alfuzosin
    CYP3A4 inhibitors
  6. Warfarin
    • Analgesics -- acetaminophen, aspirin
    • Absorption inhibitors
    • Enzyme inducers
    • Alcohol
    • HMG CoA reductase inhibitors
    • Azole antifungals
    • Cimetidine
    • Antibiotics
    • Antidepressants
    • CYP450 2C9 inhibitors
    • NSAIDs
    • Thyroid
  7. Aspirin
    Ibuprofen
  8. Antidiabetic agents:
         chlorpropamide
         glimepiride
         glipizide
         glyburide
         nateglinide
         rosiglitazone
         tolbutamide
    CYP2C9 inhibitors
  9. Antidiabetic agents:
         nateglinide
         pioglitazone
         repaglinide
         saxagliptin
         sitagliptin
    CYP3A4 inhibitors
  10. Antiarrhythmics:
         flecainide 
         mexiletine 
         propafenone
    CYP2D6 inhibitors
  11. All antidiabetic drugs
    Non-selective beta blockers
  12. Tricyclic antidepressants
    • Enzyme inducers
    • CYP2D6 inhibitors
  13. Antihypertensives:
         ACEI's
         ARB's
    NSAIDS
  14. Acetaminophen
    Enzyme inducers
  15. Non-cardioselective Beta Blockers:
         carteolol
         carvedilol
         labetalol
         levobunolol
         nadolol
         penbutolol
         pindolol
         propranolol
         sotalol
         timolol
    Epinephrine
  16. Antipsychotics:
         aripiprazole
         clozapine
         iloperidone
         lurasidone
         olanzapine
         quetiapine
         risperidone
         ziprasidone
    • Enzyme inducers 
    • Antimicrobials
    • CYP3A4 inhibitors
  17. Calcium channel blockers
    • Enzyme inducers
    • Antidepressants
    • Antimicrobials
    • 3A4 inhibitors
  18. Antidiabetic agents:
          glipizide
          glyburide
    Gastric alkalinizers
  19. Antipsychotics:
         aripiprazole
         clozapine
         iloperidone
         olanzapine
         quetiapine
         risperidone
    • Antidepressants
    • CYP2D6 inhibitors
  20. Azole antifungals:
         itraconazole 
         ketoconazole
         posaconazole
    • Gastric antisecetory agents
    • Gastric alkalinizers
  21. Antimetabolites:
         azathioprine
         mercaptopurine
    • Allopurinol
    • Febuxostat
Author
ephany
ID
169153
Card Set
ADR exam 1
Description
ADR exam 1
Updated