Antihistamines

  1. Ethanolamine
    • Diphenhydramine:
    • Tx:  anti-emetic, OTC Allergy, anti-Parkinsonism
    • ^^sedative, ^^anti-Ch
  2. Ethylaminidiamines
    • Pyrilamine:
    • ^sedative, GI side effects, ^anti-Ch
  3. Piperazines
    • Hydroxyzine:  anxiolytic
    • Cyclizine:  anti-emetic
    • Meclizine:  anti-emetic
    • ^sedate
  4. Alkylamines
    • Brompheniramine
    • Chlorpheniramine
    • Tx:  OTC Cold Rx
    • sadate, anti-Ch
  5. Phenothiazines
    • Promethazine
    • Tx:  anti-emetic
    • ^^sedative, ^^anti-Ch
  6. Cyproheptadine
    • Blocks 5-HT 2A, Musc, and H1
    • Tx:  Carcinoid Syndrome, Serotonin Syndrome (SSRI+ 5-HT agonist), Cold-induced Urticaria
  7. Loratadine
    • Claritin
    • 2nd Gen:
    • Tx:  Allergic rxt, Urticaria, Hay Fever, Insect Bites, Rx sensitivity
    • Metab by CYP3A4
  8. Cetirizine
    • Zyrtec
    • 2nd Gen
    • Tx:  Allergic Rxt, Hay Fever, Urticaria, Insect bites, Rx sensitivity
    • Metab via CYP3A4
  9. Fexofenadine
    • Allegra
    • 2nd Gen
    • Tx:  Allergic Rxt, Urticaria, Hay Fever, Insect Bite, Rx sensitivity 
    • Metab via CYP3A4
Author
emac0408
ID
167716
Card Set
Antihistamines
Description
Antihistamines
Updated