-
Benzothiadiazines
- Hydrochlorothiazide
- Chlothialidone
- SE: hypokalemia, ED, Gout, tachycardia or cardiac death (loss of K+), increased LDL, cholesterol, glucose tolerance
-
Loop diuretics
- Furosemide- good for edema
- Amiloride- K sparing
-
B-adrenergic R antagonist
ADR: Asthma, Kiabetes, SA or AV nodal dysfunction, lipid changes, rebound hypertension
-
Alpha1- adrenergic R antagonists
- Prazosin
- Terazosin
- Doxazosin
- SE: NaCl and water retention
-
Mixed Alpha/Beta R antagonist
-
NE substitute for Hypertension
- Methyldopa- metabolite active
- SE: Sedation, Depression, Dry mouth, Parkinsonian like symptoms, hepatotoxicity
-
Alpha-2 Agonist
- Clonidine
- Guanabenz
- Guanfacine
- SE: seation, xerostomia, ED, HypoT, Nightmares
-
Vesicular catecholamine transporter (VMAT2)
Reserpine- prevents storing NE and DA
-
Dihydropyridines (for HT)
- Ca++ channel Antagonists
- Amlodipine
- Nifedipine
- Verapamil
- SE: peripheral edema, GERD,
-
Cholinergic Agonists
- Bethanechol
- Methacholine
- Carbochol
- Pilocarpine
- Cevimeline
- Muscarine, Arecolin
-
Cholinergic Antagonists
- Atropine and Scopolamine
- Pirenzepine and telensepine
- ipratropium and tiotropium
- Propatheline and oxybutynin
- Benztropine mesylate, tropicamide, diclyclomine,
- Darifenacin, Solifenacin, Fesoterodine
-
Acetylcholinesterase Inhibitors
- Neostigmine, physostigmine, pyridostigmine (MG)
- Donepezil, Galantamine, Rivastigmine (Alzheimer's)
- Diisopropyl flurophosphate, isoflurophate, ecothiophate (glaucoma)
-
Nicotinic Agonists
- Nicotine
- Varenicline
- Lobeline
-
Neuromuscular Blocking Agents
- Curare, Pancuronium (competative inhibitors)
- tubocurarine, Mivacurium, atracurium, Rocuronium, Gallamine (competitive paralytics)
- Decamethonium (agonist)
- Succinylcholine (depolarizing paralytics)
- Botulinum Toxin (Ach release inhibitor)"Botox"
-
Alpha-1 Agonist
- Phenylephrine
- Mephenterimine
- Metaraminol
- Midodrine
-
Alpha-2 Agonists
- Clonidine
- Apraclonidine
- Guanfacine and Guanabenz
- Methyldopa
- Tizanidine
-
Non-Selective Alpha Agonists
- Pseudoephredrine
- Propylhexedrine
- xylometazoline
- oxymetazoline
- Naphazoline
-
Non-Selective Adrenergic Agonists
- Epinephrine
- Ephedrine
- Dopamine
-
Alpha-1 Antagonists
- Prazosin
- Terazosin
- Doxazosin
- Indoramin
- Tamsulosin, Alfuzosin, Silodosin
-
Alpha-2 Antagonist
Yohimbine
-
Non-Selective Alpha Antagonist
- Phentolamine
- Phenoxybenzamine
-
Beta-1 Antagonist
- Metoprolol
- Atenolol
- Esmolol
- Acebutolol
-
Non-Selective Beta Antagonists
- Propranolol
- Naldolol
- Timolol
- Pindolol
- Labetolol
-
Mixed Action Beta Antagonists
- Carvedilol
- Carteolol
- Betaxolol
- Celiprolol
-
Monoamine Oxidase Inhibitors
- Iproniazid (A)
- Tranylcypromine (A)
- Moclobemide (A)
- Selegiline (B)
-
Catechol-O-methyl Transferase (COMT)
-
Catecholamine Uptake Inhibitors/Releaser
- Cocaine- uptake inhibitor
- Ampehtamine, Dextro, Metha- enhance release
- Methylphenidate- enhance release
- Modafinil, Atomexatine-enhance release
- Reserpine- blocks uptake/storage to deplete Epi, NE
-
Tricyclic Anti-depressants
- Amitriptyline (5HT)
- Clomiramine (5 HT)
- Desipramine (5HT, DA)
- Nortryptyline (NE)
-
SSRI
- Citalopram
- Escitalopram
- Fluoxetine
- Paroxetine
- Sertraline
-
-
Atypical Anti-Depressants
- Buproprion (5HT, DA)
- Mirtazapine (A2 Antagonis)
- Trazodone (5HT)
-
Mood Stabilizers-Anti-convulsants
- Lithium (DA-synthesis inhibition)
- Darbamazepine, Oxcarbazepine (VG-Na-channels)
- Lamotrigine (I- glutamate release0
- Valproic Acid (increase GABA)
- Quetiapine (DA1,2, 5HT1,2)
- Aripiprazole (D23, 5HT1a,2a)
- Olanzepin (2nd gen thienobenzodiazepine)
-
H-1 antagonists (Anti-Emetics)
- Meclizine
- Cyclizine
- Diphenhydramine
- Promethazine
-
D2 Antagonists (Anti-Emetics)
- Promethazine
- Prochlorperazine
- Chlorpromazine
- Metoclopramide
- Haloperidol
- Droperidol
-
5-HT3 Antagonists (Anti-Emetics)
- Ondansetron
- Granisetron
- Dolasetron
- Palonosetron
-
CB-1 Agonist (Anti-Emetics)
Dronabinol
-
Benzodiazepines (Anti-Emetics)
-
Benzodiazepines (Sedative Hypnotics)
- Diazepam, Alprazolam, Flurazepam, Quazepam
- Temazepam and Triazolam (insomnia)
- Zolpidem, Zaleplon, Eszopiclone ( benzo-like, short acting)
-
Benzodiazepine Antagonist
Flumazenil
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