-
acetylcholine (Miochol-E)
Direct Acting Muscarinic Agonist
-
carbachol (Isopto Carbachol)
Direct Acting Muscarinic Agonist
-
methacholine (Provocholine)
Direct Acting Muscarinic Agonist
-
bethanechol (Urecholine)
Direct Acting Muscarinic Agonist
-
pilocarpine (Salagen/Ocusert Pilo)
Direct Acting Muscarinic Agonist
-
edrophonium (Tensilon)
reversible cholinesterase inhibitor
-
physostigmine/eserine
reversible cholinesterase inhibitor
-
neostigmine (Prostigmin)
reversible cholinesterase inhibitor
-
pyridostigmine (Mestinon)
reversible cholinesterase inhibitor
-
rivastigmine (Exelon)
reversible cholinesterase inhibitor
-
donepezil (Aricept)
reversible cholinesterase inhibitor
-
carbamate insecticides (e.g. Carbaryl)
reversible cholinesterase inhibitor
-
DFP/diisopropylfurophosphate/isoflurophate and echothisophate
irreversible cholinesterase inhibitor
-
organophosphate insecticides (e.g. Parathion, Malathion)
irreversible cholinesterase inhibitor
-
nerve gases used in chemical warfare (e.g. Sarin)
irreversible cholinesterase inhibitor
-
sildenafil (Viagra)
- cGMP phosphodiesterase
- (PDE-5) inhibitor
-
vardenafil (Levitra)
- cGMP phosphodiesterase
- (PDE-5) inhibitor
-
tadalafil (Cialis)
- cGMP phosphodiesterase
- (PDE-5) inhibitor
-
pralidoxime/2-PAM (Protopam)
cholinesterase reactivator
-
botulinum toxin (BOTOX)
toxin
(proteolytically degrades the SNAP-25 protein, a type of SNARE protein that is required for vesicle fusion and therefore release of ACh from presynaptic cholinergic neurons into the synaptic cleft)
-
atropine, hyoscyamine, and homatropine
Muscarinic Antagonist (Anticholinergic)
-
scopolamine and methscopolamine
Muscarinic Antagonist (Anticholinergic)
-
dicyclomine (Bentyl)
Muscarinic Antagonist (Anticholinergic)
-
propantheline
Muscarinic Antagonist (Anticholinergic)
-
glycopyrrolate (Robinul)
Muscarinic Antagonist (Anticholinergic)
-
ipratropium (Atrovent)
Muscarinic Antagonist (Anticholinergic)
-
tiatropium (Spiriva)
Muscarinic Antagonist (Anticholinergic)
-
benztropine (Cogentin)
Muscarinic Antagonist (Anticholinergic)
-
trihexyphenidyl (Artane)
Muscarinic Antagonist (Anticholinergic)
-
tolterodine (Detrol)
Muscarinic Antagonist (Anticholinergic)
-
oxybutynin (Ditropan)
Muscarinic Antagonist (Anticholinergic)
-
solifenacin (VESIcare)
Muscarinic Antagonist (Anticholinergic)
-
tropicamide (Mydriacyl)
Muscarinic Antagonist (Anticholinergic)
-
epinephrine (Adrenalin, EpiPen, Primatene Mist); E
Mixed or nonselective agonist
(?1 ≈ ?2 ≈ β1≈ β2)
-
norepinephrine (Levophed); NE
Mixed or nonselective agonist
(?1 ≈ ?2 ≈ β1>>β2)
-
isoproterenol (Isuprel)
Mixed or nonselective agonist
(β1≈ β2>> all others)
-
dopamine (Intropin); DA
Mixed or nonselective agonist
(D receptors > β1 > ?1 >> all others)
-
dobutamine (Dobutrex)
Selective β1-agonist
-
albuterol (Proventil)
Selective β2-agonist
-
metaproterenol
Selective β2-agonist
-
pirbuterol (Maxair)
Selective β2-agonist
-
salmeterol (Serevent)
Selective β2-agonist
-
terbutaline
Selective β2-agonist
-
phenylephrine
Selective ?1-agonist
-
midodrine (ProAmatine)
Selective ?1-agonist
-
cocaine
Indirect-acting sympathomimetic
-
pseudoephedrine (Sudafed)
ephedrine
Indirect-acting sympathomimetic
-
amphetamine
methamphetamine
Indirect-acting sympathomimetic
-
methylphenidate (Ritalin)
Indirect-acting sympathomimetic
-
phenytoin (Dilantin)
Traditional Antiepileptic
Blocks voltage-gated Na+ channels on neuronal axons
-
carbamazepine (Tegretol, Carbatrol)
Traditional Antiepileptic
Blocks voltage-gated Na+ channels on neuronal axons
-
ethosuximide (Zarontin)
Traditional Antiepileptic
Blocks T-type Ca2+ channels located on the postsynaptic membrane
-
valproic acid/valproate (Depakote, Depakene)
Traditional Antiepileptic/Antiseizure drug (Treatment for migraines and other headaches)
Blocks voltage-gated Na+ channels on neuronal axons
Blocks T-type Ca2+ channels located on the postsynaptic membrane
-
benzodiazepines, e.g.:
clonazepam (Klonopin)
clorazepate (Tranxene-SD)
Traditional Antiepileptic
Increase GABA effects at GABAA post-synaptic receptor
-
fosphenytoin (Cerebyx)
Traditional Antiepileptic
-
gabapentin (Neurontin)
Newer Antiepileptic/Antiseizure drug (Treatment for migraines and other headaches)
-
oxcarbazepine (Trileptal)
Newer Antiepileptic
Blocks voltage-gated Na+ channels on neuronal axons
-
lamotrigine (Lamictal)
Newer Antiepileptic
-
levetiracetam (Keppra)
Newer Antiepileptic
-
ergotamine tartrate (Ergomar)
Ergot alkaloid (Treatment for migraines and other headaches)
-
dihydroergotamine (D.H.E. 45)
Ergot alkaloid (Treatment for migraines and other headaches)
-
methysergide maleate (Sansert)
Serotonin antagonist (Treatment for migraines and other headaches)
-
sumatriptan (Imitrex)
First generation specific 5-HT1B/1D agonist (Treatment for migraines and other headaches)
-
zolmitriptan (Zomig, Zomig ZMT)
Second generation specific 5-HT1B/1D agonist (Treatment for migraines and other headaches)
-
metoclopramide (Reglan)
Dopamine antagonist (Antiemetic)
-
prochlorperazine (Compazine)
Dopamine antagonist (Antiemetic)
Relieves headache headache pain also
-
midrin (Isometheptene 65 mg + dichloralphenazone 100 mg + acetaminophen 325 mg)
Analgesic (Treatment for migraines and other headaches)
-
amitriptyline (Elavil)
Tri-cyclic antidepressant (Treatment for migraines and other headaches)
-
topiramate (Topamax)
Antiseizure drug (Treatment for migraines and other headaches)
-
morphine
Strong analgesic (µ agonist)
-
codeine
Strong analgesic (µ agonist)
-
fentanyl
Strong analgesic (µ agonist)
-
heroin
Strong analgesic (µ agonist)
-
hydrocodone (Vicodin, Lortab, Norco, others)
Strong analgesic (µ agonist)
-
hydromorphone (Dilaudid)
Strong analgesic (µ agonist)
-
meperidine (Demerol)
Strong analgesic (µ agonist)
-
methadone (Dolophine)
Strong analgesic (µ agonist)
-
oxycodone (Percodan, Percocet, OxyContin)
Strong analgesic (µ agonist)
-
propoxyphene (Darvon, Darvocet)
Strong analgesic (µ agonist)
-
pentazocine (Talwin)
Partial agonist and mixed agonist/antagonist analgesic
-
buprenorphine (Buprenex, Sabutrex, Suboxone)
Partial agonist and mixed agonist/antagonist analgesic
-
butorphanol (Stadol)
Partial agonist and mixed agonist/antagonist analgesic
-
tramadol (Ultram)
Partial agonist and mixed agonist/antagonist analgesic
-
naloxone (Narcan)
Opioid antagonist
-
naltrexone (ReVia)
Opioid antagonist
-
methylnaltrexone (Relistor)
Opioid antagonist
-
acetazolamide (Diamox)
Carbonic anhydrase inhibitor
-
mannitol (Osmitrol)
Osmotic diuretic
-
furosemide (Lasix)
- Loop diuretic/High-ceiling diuretic
- (Inhibitors of apical Na+/K+/2Cl- symport)
-
ethacrynic acid (Edecrin)
- Loop diuretic/High-ceiling diuretic
- (Inhibitors of apical Na+/K+/2Cl- symport)
-
hydrochlorothiazide (Esidrix, Hydrodiuril)
Thiazide diuretic (inhibitor of apical Na+/Cl- symport)
-
chlorothiazide (Diuril)
Thiazide diuretic (inhibitor of apical Na+/Cl- symport)
-
chlorthalidone (Hygroton)
Thiazide-like diuretic (inhibitor of apical Na+/Cl- symport)
-
indapamide (Lozol)
Thiazide-like diuretic (inhibitor of apical Na+/Cl- symport)
-
triamterene (Dyrenium)
K+ sparing diuretic (inhibitor of renal Na+ channels)
-
amiloride (Midamor)
K+ sparing diuretic (inhibitor of renal Na+ channels)
-
spironolactone (Aldactone)
K+ sparing diuretic (aldosterone antagonist)
-
eplerenone (Inspra)
K+ sparing diuretic (aldosterone antagonist)
-
drospirenone + ethinyl estradiol (Yasmin)
K+ sparing diuretic (aldosterone antagonist)
-
desmopressin acetate (1-Deamino-8-D-Arginine Vasopressin) (DDAVP, Stimate)
Anti-diuretic
-
hydrochlorothiazide (Microzide)
Thiazide diuretic (inhibitor of apical Na+/Cl- symport)
-
chlorthalidone (Thalitone)
Thiazide-like diuretic (inhibitor of apical Na+/Cl- symport)
-
reserpine
Adrenergic neuron blocker
-
methyldopa
Adrenergic neuron blocker
-
clonidine (Catapres)
Adrenergic neuron blocker
|
|